| Record Information |
| Version |
3.5 |
| Creation Date |
2005-11-16 08:48:42 -0700 |
| Update Date |
2013-02-08 17:10:44 -0700 |
| HMDB ID |
HMDB01544 |
| Secondary Accession Numbers |
None |
| Metabolite Identification |
| Common Name |
m-Chlorobenzoic acid |
| Description |
m-Chlorobenzoic acid is a metabolic byproduct of the drug bupropion. Bupropion is sold as Wellbutrin, or Zyban and is an atypical antidepressant that acts as a norepinephrine and dopamine reuptake inhibitor, and nicotinic antagonist. In 2007 it was the fourth-most prescribed antidepressant in the United States retail market, with 20.184 million retail prescriptions. |
| Structure |
Download:
MOL |
SDF |
SMILES |
InChI
Display:
2D Structure |
3D Structure
|
| Synonyms |
- 3-Cholro-benzoate
- 3-Cholro-benzoic acid
- m-Chlorobenzoate
- m-Chlorobenzoic acid
|
| Chemical Formula |
C7H5ClO2 |
| Average Molecular Weight |
156.566 |
| Monoisotopic Molecular Weight |
155.997807111 |
| IUPAC Name |
3-chlorobenzoic acid |
| Traditional IUPAC Name |
3-chlorobenzoic acid |
| CAS Registry Number |
535-80-8 |
| SMILES |
OC(=O)C1=CC(Cl)=CC=C1 |
| InChI Identifier |
InChI=1S/C7H5ClO2/c8-6-3-1-2-5(4-6)7(9)10/h1-4H,(H,9,10) |
| InChI Key |
LULAYUGMBFYYEX-UHFFFAOYSA-N |
| Chemical Taxonomy |
| Kingdom |
Organic Compounds |
| Super Class |
Aromatic Homomonocyclic Compounds |
| Class |
Benzoic Acid and Derivatives |
| Sub Class |
N/A |
| Other Descriptors |
- Organic Compounds
- monochlorobenzoic acid(ChEBI)
|
| Substituents |
- Aryl Chloride
- Benzoyl
- Carboxylic Acid
- Chlorobenzene
- Organochloride
|
| Direct Parent |
Benzoic Acid and Derivatives |
| Ontology |
| Status |
Detected and Quantified |
| Origin |
|
| Biofunction |
Not Available
|
| Application |
Not Available
|
| Cellular locations |
- Membrane (predicted from logP)
|
| Physical Properties |
| State |
Solid |
| Experimental Properties |
| Property |
Value |
Reference |
| Melting Point |
158 °C |
Not Available |
| Boiling Point |
Not Available |
Not Available |
| Water Solubility |
0.45 mg/mL |
Not Available |
| LogP |
2.68 |
HANSCH,C ET AL. (1995) |
|
| Predicted Properties |
|
| Spectra |
|
|
| Biological Properties |
| Cellular Locations |
- Membrane (predicted from logP)
|
| Biofluid Locations |
|
| Tissue Location |
Not Available
|
| Pathways |
Not Available
|
| Normal Concentrations |
|
| Urine |
Detected but not Quantified |
|
Not Applicable |
Adult (>18 years old) |
Both |
Normal
|
|
| Urine |
Detected and Quantified |
|
0.68 umol/mmol creatinine |
Adult (>18 years old) |
Both |
Normal
|
|
|
| Abnormal Concentrations |
|
Not Available |
| Associated Disorders and Diseases |
| Disease References |
None |
| Associated OMIM IDs |
None |
| External Links |
| DrugBank ID |
Not Available |
| DrugBank Metabolite ID |
Not Available |
| Phenol Explorer Compound ID |
Not Available |
| Phenol Explorer Metabolite ID |
Not Available |
| FoodDB ID |
FDB022682 |
| KNApSAcK ID |
Not Available |
| Chemspider ID |
434  |
| KEGG Compound ID |
Not Available |
| BioCyc ID |
CPD-3486  |
| BiGG ID |
Not Available |
| Wikipedia Link |
Not Available |
| NuGOwiki Link |
HMDB01544  |
| Metagene Link |
HMDB01544  |
| METLIN ID |
6311  |
| PubChem Compound |
447  |
| PDB ID |
3BZ  |
| ChEBI ID |
19985  |
| References |
| Synthesis Reference |
Wu, Wenliang; Zhu, Xurong; Zhu, Ningdong; Chen, Mingde. Methods for preparation of m-chlorobenzoic acid. Nanjing Huagong Daxue Xuebao (1997), 19(4), 117-124. |
| Material Safety Data Sheet (MSDS) |
Download (PDF)
|
| General References |
- Welch RM, Lai AA, Schroeder DH: Pharmacological significance of the species differences in bupropion metabolism. Xenobiotica. 1987 Mar;17(3):287-98.
Pubmed: 3107223
|