HMDB0000713 | Isoallolithocholic acid | 2276-93-9 | | C24H40O3 | 376.5726 376.297745146 | Not Available |
HMDB0000733 | Hyodeoxycholic acid | 83-49-8 | | C24H40O4 | 392.572 392.292659768 | Not Available |
HMDB0000760 | Hyocholic acid | 547-75-1 | | C24H40O5 | 408.5714 408.28757439 | Not Available |
HMDB0002497 | Glycochenodeoxycholate-3-sulfate | 67030-54-0 | | C26H43NO8S | 529.687 529.270938047 | Not Available |
HMDB0015151 | Glyburide | 10238-21-8 | | C23H28ClN3O5S | 494.004 493.143819418 | - Stieger B, Fattinger K, Madon J, Kullak-Ublick GA, Meier PJ: Drug- and estrogen-induced cholestasis through inhibition of the hepatocellular bile salt export pump (Bsep) of rat liver. Gastroenterology. 2000 Feb;118(2):422-30. [PubMed:10648470 ]
- Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
- Byrne JA, Strautnieks SS, Mieli-Vergani G, Higgins CF, Linton KJ, Thompson RJ: The human bile salt export pump: characterization of substrate specificity and identification of inhibitors. Gastroenterology. 2002 Nov;123(5):1649-58. [PubMed:12404239 ]
- Kemp DC, Brouwer KL: Viability assessment in sandwich-cultured rat hepatocytes after xenobiotic exposure. Toxicol In Vitro. 2004 Dec;18(6):869-77. [PubMed:15465654 ]
- Horikawa M, Kato Y, Tyson CA, Sugiyama Y: Potential cholestatic activity of various therapeutic agents assessed by bile canalicular membrane vesicles isolated from rats and humans. Drug Metab Pharmacokinet. 2003;18(1):16-22. [PubMed:15618715 ]
- Noe J, Hagenbuch B, Meier PJ, St-Pierre MV: Characterization of the mouse bile salt export pump overexpressed in the baculovirus system. Hepatology. 2001 May;33(5):1223-31. [PubMed:11343252 ]
- Funk C, Pantze M, Jehle L, Ponelle C, Scheuermann G, Lazendic M, Gasser R: Troglitazone-induced intrahepatic cholestasis by an interference with the hepatobiliary export of bile acids in male and female rats. Correlation with the gender difference in troglitazone sulfate formation and the inhibition of the canalicular bile salt export pump (Bsep) by troglitazone and troglitazone sulfate. Toxicology. 2001 Oct 5;167(1):83-98. [PubMed:11557132 ]
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HMDB0015570 | Fusidic Acid | 6990-06-3 | | C31H48O6 | 516.7092 516.345089268 | - Bode KA, Donner MG, Leier I, Keppler D: Inhibition of transport across the hepatocyte canalicular membrane by the antibiotic fusidate. Biochem Pharmacol. 2002 Jul 1;64(1):151-8. [PubMed:12106615 ]
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HMDB0014831 | Fluorescein | 2321-07-5 | | C20H12O5 | 332.3063 332.068473494 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
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HMDB0015132 | Doxorubicin | 23214-92-8 | | C27H29NO11 | 543.5193 543.174060775 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
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HMDB0015364 | Dexamethasone | 50-02-2 | | C22H29FO5 | 392.4611 392.199902243 | - Fardel O, Payen L, Courtois A, Vernhet L, Lecureur V: Regulation of biliary drug efflux pump expression by hormones and xenobiotics. Toxicology. 2001 Oct 5;167(1):37-46. [PubMed:11557128 ]
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HMDB0000659 | Deoxycholic acid disulfate | 67030-51-7 | | C24H40O10S2 | 552.698 552.20628888 | Not Available |
HMDB0000626 | Deoxycholic acid | 83-44-3 | | C24H40O4 | 392.572 392.292659768 | - Schuetz EG, Strom S, Yasuda K, Lecureur V, Assem M, Brimer C, Lamba J, Kim RB, Ramachandran V, Komoroski BJ, Venkataramanan R, Cai H, Sinal CJ, Gonzalez FJ, Schuetz JD: Disrupted bile acid homeostasis reveals an unexpected interaction among nuclear hormone receptors, transporters, and cytochrome P450. J Biol Chem. 2001 Oct 19;276(42):39411-8. Epub 2001 Aug 16. [PubMed:11509573 ]
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HMDB0014832 | Daunorubicin | 20830-81-3 | | C27H29NO10 | 527.5199 527.179146153 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
- Lecureur V, Sun D, Hargrove P, Schuetz EG, Kim RB, Lan LB, Schuetz JD: Cloning and expression of murine sister of P-glycoprotein reveals a more discriminating transporter than MDR1/P-glycoprotein. Mol Pharmacol. 2000 Jan;57(1):24-35. [PubMed:10617675 ]
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HMDB0000601 | Coprocholic acid | 547-98-8 | | C27H46O5 | 450.6511 450.334524582 | Not Available |
HMDB0014983 | Clofazimine | 2030-63-9 | | C27H22Cl2N4 | 473.396 472.122152138 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
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HMDB0014644 | Cimetidine | 51481-61-9 | | C10H16N6S | 252.339 252.115715232 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
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HMDB0000619 | Cholic acid | 81-25-4 | | C24H40O5 | 408.5714 408.28757439 | - Green RM, Hoda F, Ward KL: Molecular cloning and characterization of the murine bile salt export pump. Gene. 2000 Jan 4;241(1):117-23. [PubMed:10607905 ]
- Mita S, Suzuki H, Akita H, Stieger B, Meier PJ, Hofmann AF, Sugiyama Y: Vectorial transport of bile salts across MDCK cells expressing both rat Na+-taurocholate cotransporting polypeptide and rat bile salt export pump. Am J Physiol Gastrointest Liver Physiol. 2005 Jan;288(1):G159-67. Epub 2004 Aug 5. [PubMed:15297262 ]
- Hartmann G, Cheung AK, Piquette-Miller M: Inflammatory cytokines, but not bile acids, regulate expression of murine hepatic anion transporters in endotoxemia. J Pharmacol Exp Ther. 2002 Oct;303(1):273-81. [PubMed:12235261 ]
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HMDB0014620 | Chlorpromazine | 50-53-3 | | C17H19ClN2S | 318.864 318.095747015 | - Wang EJ, Casciano CN, Clement RP, Johnson WW: Fluorescent substrates of sister-P-glycoprotein (BSEP) evaluated as markers of active transport and inhibition: evidence for contingent unequal binding sites. Pharm Res. 2003 Apr;20(4):537-44. [PubMed:12739759 ]
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HMDB0006898 | Chenodeoxyglycocholic acid | | | C26H43NO5 | 449.6233 449.314123491 | Not Available |
HMDB0002522 | Chenodeoxycholic acid sulfate | 59132-31-9 | | C24H40O7S | 472.635 472.249474324 | Not Available |
HMDB0000545 | Chenodeoxycholic acid disulfate | 60262-91-1 | | C24H40O10S2 | 552.698 552.20628888 | Not Available |
HMDB0002586 | Chenodeoxycholic acid 3-sulfate | 59132-32-0 | | C24H40O7S | 472.635 472.249474324 | Not Available |
HMDB0000518 | Chenodeoxycholic acid | 474-25-9 | | C24H40O4 | 392.572 392.292659768 | Not Available |
HMDB0014699 | Bosentan | 147536-97-8 | | C27H29N5O6S | 551.614 551.183854375 | - Fattinger K, Funk C, Pantze M, Weber C, Reichen J, Stieger B, Meier PJ: The endothelin antagonist bosentan inhibits the canalicular bile salt export pump: a potential mechanism for hepatic adverse reactions. Clin Pharmacol Ther. 2001 Apr;69(4):223-31. [PubMed:11309550 ]
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HMDB0002082 | Bisnorcholic acid | | | C22H36O5 | 380.5182 380.256274262 | Not Available |
HMDB0000506 | alpha-Muricholic acid | 2393-58-0 | | C24H40O5 | 408.579 408.287574388 | Not Available |